摘要
以苯肼、乙酰乙酸乙酯和氨基杂环为原料 ,合成了两类含双杂环的新型吡唑甲酰胺衍生物 ,其结构经元素分析、1HNMR ,MS及IR确证 .初步的生物活性测试结果表明 :部分化合物对水稻纹枯病菌、小麦赤霉病菌和苹果轮纹病菌具有良好的抑制效果 .
In order to search for novel fungicides with high activity and low toxicity, a series of bis-heterocyclic compounds containing 1H-pyrazole and thiazole were designed and synthesized from phenyl hydrazine, ethyl acetoacetate and aromatic aminoheterolcycles. The structures of all new compounds were confirmed by elemental analysis, H-1 NMR, IR and MS spectra. Preliminary bioassays indicated that some compounds showed fungicidal activity against Pellicularia sasakii, Gibberella zeave and Physalospora piricola.
出处
《有机化学》
SCIE
CAS
CSCD
北大核心
2003年第10期1131-1134,共4页
Chinese Journal of Organic Chemistry
基金
科技部国家"九五"重点科技攻关 (No .97 563 0 2 0 5)资助项目
