An expedient,synthetic method to fused polycyclic derivatives of isoquinoline is described via tandem reaction of isoquinoline,dialkyl acetylenedicarboxylates and dialkyl chloromalonate.
An effective route to pyrrolo[1,2-a]pyrazines is described via reaction of ethylenediamine,acetylenic esters and nitrostyrene derivatives in the presence of 20 mol%of sulfamic acid.
A simple and efficient synthetic protocol has been developed using a one-pot multicomponent reaction (MCR) involving 2-aminophenols, dialkyl acetylenedicarboxylates, and ethyl bromopyruvate in poly(ethyleneglycol)...A simple and efficient synthetic protocol has been developed using a one-pot multicomponent reaction (MCR) involving 2-aminophenols, dialkyl acetylenedicarboxylates, and ethyl bromopyruvate in poly(ethyleneglycol). This protocol was utilized to prepare novel pyrrolo[2,1-c][1,4]benzoxazines in excellent yields.展开更多
A simple and efficient synthetic protocol has been developed using a one-pot, three-component reaction involving 2-amino phenols, dialkyl acetylene dicarboxylates and nitrostyrene derivatives. Utilizing this protocol,...A simple and efficient synthetic protocol has been developed using a one-pot, three-component reaction involving 2-amino phenols, dialkyl acetylene dicarboxylates and nitrostyrene derivatives. Utilizing this protocol, a variety of novel pyrrolo-1,4-benzoxazine derivatives were synthesized in excellent yields.展开更多
基金Sanandaj Branch, Islamic Azad University Research Council for the fnancial support of this research
文摘An expedient,synthetic method to fused polycyclic derivatives of isoquinoline is described via tandem reaction of isoquinoline,dialkyl acetylenedicarboxylates and dialkyl chloromalonate.
文摘An effective route to pyrrolo[1,2-a]pyrazines is described via reaction of ethylenediamine,acetylenic esters and nitrostyrene derivatives in the presence of 20 mol%of sulfamic acid.
基金Sanandaj Branch,Islamic Azad University Research Council for the financial support
文摘A simple and efficient synthetic protocol has been developed using a one-pot multicomponent reaction (MCR) involving 2-aminophenols, dialkyl acetylenedicarboxylates, and ethyl bromopyruvate in poly(ethyleneglycol). This protocol was utilized to prepare novel pyrrolo[2,1-c][1,4]benzoxazines in excellent yields.
文摘A simple and efficient synthetic protocol has been developed using a one-pot, three-component reaction involving 2-amino phenols, dialkyl acetylene dicarboxylates and nitrostyrene derivatives. Utilizing this protocol, a variety of novel pyrrolo-1,4-benzoxazine derivatives were synthesized in excellent yields.